Resumes
Resumes
John Stellwagen Phones & Addresses
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Newbury Park, CA
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12 Elnew Ave, Beverly, MA 01915 (978) 922-4941
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1409 Cedar St, Iowa City, IA 52245 (319) 338-6495
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918 Prologue Rd, Durham, NC 27712
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Sherman Oaks, CA
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Valley Village, CA
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Pasadena, CA
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El Cerrito, CA
Publications
Us Patents
Benzene Sulfonamide Thiazole And Oxazole Compounds
View pageUS Patent:
20090298815, Dec 3, 2009
Filed:
May 4, 2009
Appl. No.:
12/434963
Inventors:
Jerry Leroy Adams - Collegeville PA, US
Scott Howard Dickerson - Durham NC, US
Neil W. Johnson - Collegeville PA, US
Kevin Kuntz - Durham NC, US
Kimberly Petrov - Durham NC, US
Jeffrey M. Ralph - Collegeville PA, US
Tara Renae Rheault - Durham NC, US
Gregory Schaaf - Durham NC, US
John Stellwagen - Durham NC, US
Xinrong Tian - Collegeville PA, US
David Edward Uehling - Durham NC, US
Alex Gregory Waterson - Durham NC, US
Brian Wilson - Durham NC, US
Scott Howard Dickerson - Durham NC, US
Neil W. Johnson - Collegeville PA, US
Kevin Kuntz - Durham NC, US
Kimberly Petrov - Durham NC, US
Jeffrey M. Ralph - Collegeville PA, US
Tara Renae Rheault - Durham NC, US
Gregory Schaaf - Durham NC, US
John Stellwagen - Durham NC, US
Xinrong Tian - Collegeville PA, US
David Edward Uehling - Durham NC, US
Alex Gregory Waterson - Durham NC, US
Brian Wilson - Durham NC, US
International Classification:
A61K 31/506
C07D 417/04
C07D 417/14
A61K 31/5377
A61K 31/541
A61P 35/00
C07D 417/04
C07D 417/14
A61K 31/5377
A61K 31/541
A61P 35/00
US Classification:
5142278, 544331, 544122, 544295, 544 582, 514275, 5142358, 51425219
Abstract:
The present invention provides thiazole sulfonamide and oxazole sulfonamide compounds, compositions containing the same, as well as processes for the preparation and methods for their use as pharmaceutical agents.
Benzene Sulfonamide Thiazole And Oxazole Compounds
View pageUS Patent:
20110172215, Jul 14, 2011
Filed:
May 4, 2009
Appl. No.:
12/991004
Inventors:
George Adjabeng - Durham NC, US
Jeffrey Leroy Adams - Collegeville PA, US
Scott Howard Dickerson - Durham NC, US
Keith Hornberger - Mount Sinai NY, US
Neil W. Johnson - Collegeville PA, US
Kevin Kuntz - Durham NC, US
Kimberly Petrov - Durham NC, US
Jeffrey M. Ralph - Collgeville PA, US
Tara Renae Rheault - Durham NC, US
Gregory Schaaf - Durham NC, US
John Stellwagen - Durham NC, US
Xinrong Tian - Collegeville NC, US
David E. Uehling - Durham NC, US
Alex G. Waterson - Durham NC, US
Brian Wilson - Durham NC, US
Jeffrey Leroy Adams - Collegeville PA, US
Scott Howard Dickerson - Durham NC, US
Keith Hornberger - Mount Sinai NY, US
Neil W. Johnson - Collegeville PA, US
Kevin Kuntz - Durham NC, US
Kimberly Petrov - Durham NC, US
Jeffrey M. Ralph - Collgeville PA, US
Tara Renae Rheault - Durham NC, US
Gregory Schaaf - Durham NC, US
John Stellwagen - Durham NC, US
Xinrong Tian - Collegeville NC, US
David E. Uehling - Durham NC, US
Alex G. Waterson - Durham NC, US
Brian Wilson - Durham NC, US
International Classification:
A61K 31/541
C07D 417/14
A61K 31/5377
A61K 31/506
C07D 413/14
C07D 417/04
A61P 35/00
C07D 417/14
A61K 31/5377
A61K 31/506
C07D 413/14
C07D 417/04
A61P 35/00
US Classification:
5142278, 544122, 5142358, 514272, 544297, 544 582, 5142322, 544107
Abstract:
The present invention provides thiazole sulfonamide and oxazole sulfonamide compounds, compositions containing the same, as well as processes for the preparation and methods for their use as pharmaceutical agents.
Thiazole And Oxazole Kinase Inhibitors
View pageUS Patent:
20110190280, Aug 4, 2011
Filed:
Aug 27, 2008
Appl. No.:
12/674016
Inventors:
George Adjabeng - Durham NC, US
Neil Bifulco - Durham NC, US
Ronda G. Davis-Ward - Durham NC, US
Scott Howard Dickerson - Durham NC, US
Kelly Horne Donaldson - Durham NC, US
Philip Anthony Harris - Wayne PA, US
Keith Hornberger - Durham NC, US
Kimberly Petrov - Durham NC, US
Tara Renae Rheault - Durham NC, US
Gregory Schaaf - Durham NC, US
John Stellwagen - Durham NC, US
David Edward Uehling - Durham NC, US
Alex Gregory Waterson - Durham NC, US
Neil Bifulco - Durham NC, US
Ronda G. Davis-Ward - Durham NC, US
Scott Howard Dickerson - Durham NC, US
Kelly Horne Donaldson - Durham NC, US
Philip Anthony Harris - Wayne PA, US
Keith Hornberger - Durham NC, US
Kimberly Petrov - Durham NC, US
Tara Renae Rheault - Durham NC, US
Gregory Schaaf - Durham NC, US
John Stellwagen - Durham NC, US
David Edward Uehling - Durham NC, US
Alex Gregory Waterson - Durham NC, US
International Classification:
A61K 31/541
C07D 403/14
A61K 31/506
C07D 413/14
A61K 31/5377
C07D 417/14
C07D 498/04
A61K 31/5365
A61P 35/00
C07D 403/14
A61K 31/506
C07D 413/14
A61K 31/5377
C07D 417/14
C07D 498/04
A61K 31/5365
A61P 35/00
US Classification:
5142278, 544295, 51425218, 544331, 514275, 544122, 5142358, 544 582, 544105, 5142305
Abstract:
The present invention provides thiazole and oxazole compounds, compositions containing the same, as well as processes for the preparation and methods for their use as pharmaceutical agents.
Heteroaryl Compounds As Pikk Inhibitors
View pageUS Patent:
20120190666, Jul 26, 2012
Filed:
May 12, 2010
Appl. No.:
13/319683
Inventors:
Christiane Bode - Somerville MA, US
Alessandro Boezio - Somerville MA, US
Alan C. Cheng - San Francisco CA, US
Deborah Choquette - Medford MA, US
James Robert Coats - Oak Harbor WA, US
Katrina Woodin Copeland - Sudbury MA, US
Hongbing Huang - Lexington MA, US
Daniel La - Brookline MA, US
Richard Thomas Lewis - Framingham MA, US
Hongyu Liao - Thousand Oaks CA, US
Michele Potashman - Cambridge MA, US
John Stellwagen - Beverly MA, US
Shuyan Yi - Cambridge MA, US
Mark H. Norman - Thousand Oaks CA, US
Markian M. Stec - Moorpark CA, US
Emily Anne Peterson - Cambridge MA, US
Russell Graceffa - Hampton NH, US
Alessandro Boezio - Somerville MA, US
Alan C. Cheng - San Francisco CA, US
Deborah Choquette - Medford MA, US
James Robert Coats - Oak Harbor WA, US
Katrina Woodin Copeland - Sudbury MA, US
Hongbing Huang - Lexington MA, US
Daniel La - Brookline MA, US
Richard Thomas Lewis - Framingham MA, US
Hongyu Liao - Thousand Oaks CA, US
Michele Potashman - Cambridge MA, US
John Stellwagen - Beverly MA, US
Shuyan Yi - Cambridge MA, US
Mark H. Norman - Thousand Oaks CA, US
Markian M. Stec - Moorpark CA, US
Emily Anne Peterson - Cambridge MA, US
Russell Graceffa - Hampton NH, US
Assignee:
Amgen Inc. - Thousand Oaks CA
International Classification:
A61K 31/52
C07D 401/14
A61K 31/506
A61P 35/02
A61K 31/53
C07D 487/04
A61K 31/5377
A61P 35/00
C07D 473/40
C07D 471/04
C07D 401/14
A61K 31/506
A61P 35/02
A61K 31/53
C07D 487/04
A61K 31/5377
A61P 35/00
C07D 473/40
C07D 471/04
US Classification:
51421021, 544264, 51426323, 544328, 514256, 544212, 514245, 544236, 514248, 544296, 544117, 5142332
Abstract:
The present invention provides compounds that are PIKK inhibitors, more specifically, mTOR and/or PI3Kα kinase inhibitors and are therefore useful for the treatment of diseases treatable by inhibition of kinases, specifically PI3 kinases, more specifically, mTOR and/or PI3Kα, such as cancer. Also provided are pharmaceutical compositions containing such compounds and processes for preparing such compounds.
Benzene Sulfonamide Thiazole And Oxazole Compounds
View pageUS Patent:
20130144055, Jun 6, 2013
Filed:
Jan 31, 2013
Appl. No.:
13/755466
Inventors:
George Adjabeng - Durham NC, US
Jerry Leroy Adams - Collegeville PA, US
Scott Howard Dickerson - Durham NC, US
Keith Hornberger - Mount Sinal NY, US
Neil W. Johnson - Collegeville PA, US
Kevin Kuntz - Durham NC, US
Kimberly Petrov - Durham NC, US
Jeffrey M. Ralph - Collegeville PA, US
Tara Renae Rheault - Durham NC, US
Gregory Schaaf - Durham NC, US
John Stellwagen - Durham NC, US
Xinrong Tian - Collegeville PA, US
David E. Uehling - Durham NC, US
Alex G. Waterson - Durham NC, US
Brian Wilson - Durham NC, US
Jerry Leroy Adams - Collegeville PA, US
Scott Howard Dickerson - Durham NC, US
Keith Hornberger - Mount Sinal NY, US
Neil W. Johnson - Collegeville PA, US
Kevin Kuntz - Durham NC, US
Kimberly Petrov - Durham NC, US
Jeffrey M. Ralph - Collegeville PA, US
Tara Renae Rheault - Durham NC, US
Gregory Schaaf - Durham NC, US
John Stellwagen - Durham NC, US
Xinrong Tian - Collegeville PA, US
David E. Uehling - Durham NC, US
Alex G. Waterson - Durham NC, US
Brian Wilson - Durham NC, US
Assignee:
GlaxoSmithKline LLC - Philadelphia PA
International Classification:
C07D 417/14
C07D 417/04
C07D 413/04
C07D 413/14
C07D 403/14
C07D 417/04
C07D 413/04
C07D 413/14
C07D 403/14
US Classification:
544 60, 544122, 544295, 544331
Abstract:
The present invention provides thiazole sulfonamide and oxazole sulfonamide compounds, compositions containing the same, as well as processes for the preparation and methods for their use as pharmaceutical agents.
Benzimidazole And Azabenzimidazole Compounds That Inhibit Anaplastic Lymphoma Kinase
View pageUS Patent:
20130217668, Aug 22, 2013
Filed:
Jul 28, 2011
Appl. No.:
13/813813
Inventors:
Christiane M. Boezio - Somerville MA, US
Alan C. Cheng - San Francisco CA, US
Deborah Choquette - Medford MA, US
Richard T. Lewis - Framingham MA, US
Michele H. Potashman - Cambridge MA, US
Karina Romero - Arlington MA, US
John C. Stellwagen - Beverly MA, US
Douglas A. Whittington - Waltham MA, US
Alan C. Cheng - San Francisco CA, US
Deborah Choquette - Medford MA, US
Richard T. Lewis - Framingham MA, US
Michele H. Potashman - Cambridge MA, US
Karina Romero - Arlington MA, US
John C. Stellwagen - Beverly MA, US
Douglas A. Whittington - Waltham MA, US
Assignee:
AMGEN INC. - Thousand Oaks CA
International Classification:
C07D 471/04
C07D 401/10
C07D 413/14
C07D 401/14
C07D 417/14
C07D 403/08
C07D 235/30
C07D 413/10
C07D 401/10
C07D 413/14
C07D 401/14
C07D 417/14
C07D 403/08
C07D 235/30
C07D 413/10
US Classification:
51421018, 546118, 5483074, 546199, 544139, 544364, 544127, 5483061, 544 582, 514303, 514388, 514322, 5142345, 51425309, 5142342, 51425304
Abstract:
Compounds of Formula (I) are useful inhibitors of anaplastic lymphoma kinase. Compounds of Formula (I) have the following structure: where the definitions of the variables are provided herein.
Benzene Sulfonamide Thiazole And Oxazole Compounds
View pageUS Patent:
20140080851, Mar 20, 2014
Filed:
Nov 25, 2013
Appl. No.:
14/088598
Inventors:
JERRY LEROY ADAMS - COLLEGEVILLE PA, US
SCOTT HOWARD DICKERSON - DURHAM NC, US
KEITH HORNBERGER - DURHAM NC, US
NEIL W. JOHNSON - COLLEGEVILLE PA, US
KEVIN KUNTZ - DURHAM NC, US
KIMBERLY PETROV - DURHAM NC, US
JEFFREY M. RALPH - COLLEGEVILLE PA, US
TARA RENAE RHEAULT - DURHAM NC, US
GREGORY SCHAAF - DURHAM NC, US
JOHN STELLWAGEN - DURHAM NC, US
XINRONG TIAN - COLLEGEVILLE PA, US
DAVID E. UEHLING - DURHAM NC, US
ALEX G. WATERSON - DURHAM NC, US
BRIAN WILSON - DURHAM NC, US
SCOTT HOWARD DICKERSON - DURHAM NC, US
KEITH HORNBERGER - DURHAM NC, US
NEIL W. JOHNSON - COLLEGEVILLE PA, US
KEVIN KUNTZ - DURHAM NC, US
KIMBERLY PETROV - DURHAM NC, US
JEFFREY M. RALPH - COLLEGEVILLE PA, US
TARA RENAE RHEAULT - DURHAM NC, US
GREGORY SCHAAF - DURHAM NC, US
JOHN STELLWAGEN - DURHAM NC, US
XINRONG TIAN - COLLEGEVILLE PA, US
DAVID E. UEHLING - DURHAM NC, US
ALEX G. WATERSON - DURHAM NC, US
BRIAN WILSON - DURHAM NC, US
Assignee:
GLAXOSMITHKLINE LLC - PHILADELPHIA PA
International Classification:
C07D 417/04
US Classification:
514275
Abstract:
The present invention provides thiazole sulfonamide and oxazole sulfonamide compounds, compositions containing the same, as well as processes for the preparation and methods for their use as pharmaceutical agents.
Cyclopropyl Dihydroquinoline Sulfonamide Compounds
View pageUS Patent:
20210387977, Dec 16, 2021
Filed:
Jun 10, 2021
Appl. No.:
17/344939
Inventors:
- Thousand Oaks CA, US
Isaac E. MARX - Arlington MA, US
John STELLWAGEN - Beverly MA, US
Wei ZHAO - Westford MA, US
Alan H. CHERNEY - Somerville MA, US
Isaac E. MARX - Arlington MA, US
John STELLWAGEN - Beverly MA, US
Wei ZHAO - Westford MA, US
Alan H. CHERNEY - Somerville MA, US
Assignee:
AMGEN INC. - THOUSAND OAKS CA
International Classification:
C07D 413/12
Abstract:
The present invention provides a compound of Formula (I):